#EXP00308

General

Accession EXP00308
Activity Formation (3-24h)
Date 2014-11-23
Administration Coated
Model in vivo
Organism Staphylococcus aureus Smith diffuse SD)
Status Validated
Notes Peptide adsorbed to Dracon graft

Peptide

FS3

YAPWTNF

Experimental activity

Method Concentration Notes
Total countable CFUs 0.65 nmol/cm2 in vivo (rat model).
Total countable CFUs 0.6 nmol/cm2 in vivo (rat model).Synergism with Daptomycin (6mg/Kg)

References

Quorum sensing inhibitor FS3-coated vascular graft enhances daptomycin efficacy in a rat model of staphylococcal infection

Oscar Cirioni, Federico Mocchegiani, Ivana Cacciatore, Jacopo Vecchiet, Carmela Silvestri, Leonardo Baldassarre, Claudio Ucciferri, Elena Orsetti, Pamela Castelli, Mauro Provinciali, Marco Vivarelli, Erika Fornasari, Andrea Giacometti

2013. Peptides :77-81